Patents

CA2961166: Alkylidene phosphonate esters as P-glycoprotein inducers

The invention relates to the alkylidene phosphonate esters of formula I wherein, R1 is selected from a group consisting of hydrogen or alkyl group; R2 is selected from a group consisting of hydrogen, hydroxy, alkyl, alkoxy, nitro, halogen, amino, N- substituted alkylamino; alkyl group is selected from a group consisting of methyl, ethyl and isopropyl; Ar is selected from a group consisting of aryl, substituted aryl, fused aryl, heteroaryl, and substituted heteroaryl. The invention particularly relates to synthesis and P-glycoprotein induction activity of the alkylidene phosphonate esters. In addition, the invention relates to methods of using compounds for treating or preventing Alzheimer's disease.

Filing Date: 13-03-2017

Issue Date: 13-03-2017

Applicant: CSIR-Indian Institute of Integrative Medicine (CSIR-IIIM), Jammu

Patent No: CA2961166

Application No: 2961166

Inventor(s): Bharate Sandip, Kumar Ajay, Manda Sudhakar, Joshi Prashant, Bharate Sonali, Wani Abubakar, Sharma Sadhana, Vishwakarma Ram

IPC Classification: A61K31/663, A61K31/665, A61P25/28, C07F9/40, C07F9/655

Country: Canada

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