Patents

IN347344: Spiro-oxazines, indolinones and preparation thereof

The invention relates to novel spiro-oxazine analogues and Indolinone compounds or positional isomers, or stereoisomers, or derivatives, or pharmaceutically acceptable salt thereof. Further, the invention provides transition-metal free Multicomponent Reaction (MCR) process for the preparation of said compounds using aryne precursor, N-substituted isatin and N-heteroaromatic compound as the nucleophile under mild conditions leading to the formation of the desired complex of spiro-oxazine analogues (I) and indolinone analogues (II) in high yield and selectivity.

Filing Date: 15-05-2013

Issue Date: 22-09-2020

Applicant: CSIR-National Chemical Laboratory (CSIR-NCL), Pune

Patent No: IN347344

Application No: 1440/DEL/2013

Inventor(s): Akkattu, Thankappan Biju; Anup Bhunia; Tony Roy

IPC Classification: C07D

Country: India

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