Patents

IN356367: 2-benzyl-indanone compounds as anticancer agent and a process for preparation thereof

The anticancer activity of gallic acid compounds has been invented, in order to obtain new potent and cost effective molecule using in vitro cytotoxicity assay. The invention particularly relates to the gallic acid based new molecules i.e. 2-benzyl indanones represented by structure 1, possessing anticancer activity against human cancer cell lines. The compound also exhibited tubulin polymerisation inhibition. 2-(3',4'-methylenedioxybenzyl)-3-(3",4",5"-trimethoxyphenyl)-indanone- 1 (2), possessing molecular formulae as C29H30O9 was synthesized from gallic acid, exhibits potent in-vivo anticancer activity. Compound 2 was evaluated for acute oral activity in Swiss albino mice and it was found to be well tolerated by the experimental animals up to 300mg/kg body weight. (Formula 1, Formula 2).

Filing Date: 13-07-2015

Issue Date: 21-01-2021

Applicant: CSIR-Central Institute of medicinal and Aromatic Plants (CSIR-CIMAP), Lucknow

Patent No: IN356367

Application No: 2105DEL2015

Inventor(s): Arvind Singh Negi, Aastha Singh, Suaid Luqman, Debabrata Chanda, Dilip Manikrao Mondhe, Ajit Kumar Saxena, Kaneez Fatima, Arjun Singh

Country: India

Related Patents